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Cat. No. Product Name Target Signaling Pathways
T12477 Uzansertib phosphate

INCB053914 phosphate

Pim Chromatin/Epigenetic; JAK/STAT signaling
Uzansertib phosphate (INCB053914 phosphate) 是一种可口服的 ATP 竞争性泛-PIM 激酶抑制剂,对多种血液肿瘤细胞系具有广泛的抗增殖活性,对 PIM1、PIM2 和 PIM3 的 IC50分别为 0.24 、30 和 0.12 nM。
T39090 Uzansertib

INCB053914

Uzansertib (INCB053914) is a potent ATP-competitive pan-PIM kinase inhibitor. It exhibits exceptional inhibitory activity against PIM1, PIM2, and PIM3 with IC50 values of 0.24 nM, 30 nM, and 0.12 nM, respectively. Furthermore, Uzansertib demonstrates significant anti-proliferative effects against an assorted range of hematologic tumor cell lines.

化合物

Uzansertib phosphate
Cat.No: T12477
Synonym: INCB053914 phosphate
Target: Pim
Uzansertib
Cat.No: T39090
Synonym: INCB053914
Target:
TargetMol Loading
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